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21.06.2002 US 390874P
(54) CIS-2,4,5- TRIPHENYL-IMIDAZOLINE UND IHRE
VERWENDUNG BEI DER BEHANDLUNG VON
TUMOREN
(73)F.HOFFMANN-LA ROCHE AG
Grenzacherstrasse124
4070 Basel (CH)
(72)LIU, Emily,Aijun
191 AlexanderAvenue
Nutley,NJ07110(US)
KONG, Norman
12KlimbackCourt
West Caldwell,NJ07006 (US)
VU, Binh,Thanh
1WillowLane
NorthCaldwell,NJ07006 (US)
(86)PCT/EP 2002/013904(en)
(87)WO 2003/051359 26.6.2003
(51) A61K0031/4178 (2006.01) Z C07 D0405/06 (2006.01)
(11) 01473 293
(51) A61K0031/4184 (2006.01) Z A61K0031/4545
(2006.01)
(11) 01499 316
(51) A61K0031/422 (2006.01) Z A61K0031/4164
(2006.01)
(11) 01458 380
(51) A61K0031/425 (2006.01)
A61K0047/12 (2006.01)
A61K0047/02 (2006.01)
A61P0035/00 (2006.01)
(11) 01353668
(21) 02713446.9
(22)22.01.2002 (86)en
(43)22.10.2003 (87)en
(24) 19.03.2008
(30)25.01.2001US 264228P
11.05.2001US 290008P
(54) VERFAHREN ZUR HERSTELLUNG VON
PHARMAZEUTISCHEN ZUSAMMENSETZUNGEN
ENTHALTEND EPOTHILON-ANALOGA ZUR
KREBSBEHANDLUNG
(73)Bristol-Myers Squibb Company
P.O.Box4000,Lawrenceville-Princeton Road
Princeton,NJ08543(US)
(72)MALLOY, Timothy,M.
1902 Makefield Rd.
Yardley,PA19067 (US)
RAGHAVAN, Krishnaswamy,Srinivas
3Hickory Ct.
Cranbury,NJ08512(US)
VARIA, Sailesh,Amilal
10Claredon Ct.
Princeton Junction,NJ08550(US)
BANDYOPADHYAY, Rebanta
7492CapriSt
Portage,MI49002 (US)
PANAGGIO, Andrea
5Tindall Trail
West Windsor,NJ08505(US)
(86)PCT/US 2002/001813(en)
(87)WO 2002/058700 1.8.2002
(51) A61K0031/428 (2006.01) Z C07 D0417/14 (2006.01)
(11) 01636 223
(51) A61K0031/437 (2006.01)
A61K0009/16 (2006.01)
A61K0047/14 (2006.01)
A61K0047/44 (2006.01)
A61K0009/00 (2006.01)
A61P0025/20 (2006.01)
(11) 01469848
(21) 03729537.5
(22)09.01.2003 (86)en
(43)27.10.2004(87)en
(24) 19.03.2008
(30)10.01.2002 US 346613P
(54) SEDIERENDE
NICHT-BENZODIAZEPIN-FORMULIERUNGEN
(73)BIOVAIL LABORATORIES INTERNATIONAL SRL
Chelston ParkBuilding 2,
CollymoreRockSaintMichael (BB)
(72)OTOOLE, Edel
70 Philipsburgh Terrace,Marino
(51) A61K0031/444 (2006.01) Z C07 D0401/12 (2006.01)
(11) 01562 933
(51) A61K0031/445 (2006.01) Z A61K0039/04 (2006.01)
(11) 00 971735
(51) A61K0031/445 (2006.01) Z C07 C0069/738 (2006.01)
(11) 01307 423
(51) A61K0031/445 (2006.01) Z C07 D0211/46 (2006.01)
(11) 01362 031
(51) A61K0031/445 (2006.01)
A61P0037/08 (2006.01)
C07 D0211/22 (2006.01)
(11) 01414 453
(21) 02751479.3
(22)29.07.2002 (86)en
(43)06.05.2004(87)en
(24) 19.03.2008
(30)31.07.2001EP 01610081
(54) FEXOFENADINE HYDROCHLORID POLYMORPH
(73)TexcontorEtablissement
Heiligkreuz 40,
Postfach39
9490Vaduz (LI)
(72)MILLA, FredericoJunquera
C/CineastaAdolfo AznarNo.3,Esc.1a, 4.,B.
50015 Zaragoza(ES)
(86)PCT/IB 2002/002954 (en)
(87)WO 2003/011295 13.2.2003
(51) A61K0031/454 (2006.01) Z A61K0031/4164
(2006.01)
(11) 01458 380
(51) A61K0031/4545 (2006.01) Z A61K0031/4164
(2006.01)
(11) 01458 380
(51) A61K0031/4545 (2006.01)
C07 D0471/04 (2006.01)
C07 D0401/14 (2006.01)
A61K0031/4184 (2006.01)
A61P0037/08 (2006.01)
(11) 01499 316
(21) 03719766.2
(22)16.04.2003 (86)en
(43)26.01.2005(87)en
(24) 19.03.2008
(30)18.04.2002 US 373731P
(54) 1-(4-PIPERIDINYL)BENZIMIDAZOLE ALS HISTAMIN
H3ANTAGONISTEN
(73)Schering Corporation
2000 Galloping Hill Road
Kenilworth,NewJersey07033-0530 (US)
(72)MANGIARACINA, Pietro
4MontclairAvenue
Monsey,NY10952(US)
TOM, Wing,C.
133 CedarGroveParkway
CedarGrove,NJ07009(US)
SOLOMON, Daniel,M.
9Marshall Drive
Edison,NJ08817(US)
ASLANIAN, Robert,G.
144 Philip Drive
Rockaway,NJ07866 (US)
ROSENBLUM, Stuart,B.
16Steven Terrace
West Orange,NJ07052(US)
SHIH, Neng-Yang
1Maple Drive
NorthCaldwell,NJ07006 (US)
BERLIN, Michael,Y.
14 HendrickRoad
Flemington,NJ08822 (US)
BOYCE, Christopher,W.
71Bonnell Street
Flemington,NJ08822 (US)
CAO, Jianhua
252West Locust Avenue
Edison,NJ08820 (US)
MC CORMICK, Kevin,D.
15 Brookfield Road
Basking Ridge,NJ07920 (US)
ZENG, Qingbei
509CiderRoad
Dublin 3(IE)
FOGARTY, Siobhan
88 Temple Road
Blackrock,County Dublin (IE)
(86)PCT/IE 2003/000001(en)
(87)WO 2003/059349 24.7.2003
(51) A61K0031/4375 (2006.01) Z C07 D0471/04 (2006.01)
(11) 01713804
(51) A61K0031/44 (2006.01) Z C07 D0213/74 (2006.01)
(11) 01042293
(51) A61K0031/44 (2006.01)
A61K0031/472 (2006.01)
A61K0031/47 (2006.01)
A61K0031/164 (2006.01)
A61P0031/04 (2006.01)
C07 D0471/04 (2006.01)
C07 D0213/42 (2006.01)
C07 C0239/14 (2006.01)
C07 D0217/02 (2006.01)
C07 D0215/20 (2006.01)
(11) 01283711
(21) 01935094.1
(22)04.05.2001(86)en
(43)19.02.2003 (87)en
(24) 19.03.2008
(30)05.05.2000 US 201943P
04.10.2000 US 238084 P
(54) INHIBITOREN VON PEPTID DEFORMYLASE
(73)SMITHKLINE BEECHAM CORPORATION
One Franklin PlazaP.O.Box7929
Philadelphia, PA 19101(US)
(72)AUBART, Kelly,M.
709Swedeland Road
King of Prussia, PA 19406 (US)
CHRISTENSEN, Siegfried,B.,IV
709Swedeland Road
King of Prussia, PA 19406 (US)
BRIAND, Jacques
709Swedeland Road
King of Prussia, PA 19406 (US)
CUMMINGS, Maxwell,David
659 West ValleyRoad
Strafford,PA19087(US)
(86)PCT/US 2001/014593(en)
(87)WO 2001/085170 15.11.2001
(51) A61K0031/44 (2006.01)
A61K0031/47 (2006.01)
A61K0031/53 (2006.01)
A61K0031/505 (2006.01)
C07 D0215/00 (2006.01)
C07 D0217/00 (2006.01)
C07 D0253/00 (2006.01)
C07 D0401/00 (2006.01)
C07 D0403/00 (2006.01)
C07 D0471/00 (2006.01)
C07 D0515/00 (2006.01)
A61P0025/36 (2006.01)
(11) 01363 630
(21) 02713374.3
(22)07.01.2002 (86)en
(43)26.11.2003 (87)en
(24) 19.03.2008
(30)08.01.2001US 755021
(54) KAPPA-OPIOID-REZEPTOR-LIGANDEN
(73)RESEARCH TRIANGLE INSTITUTE
3040CornwallisRoad,P.O.Box12194
ResearchTriangle Park,NC27709(US)
(72)THOMAS, James,B.
3620 RabbitHill Lane
Efland,NC27243(US)
MASCARELLA, S.,Wayne
1823 Borland Road
Hillsborough,NC27278(US)
CARROLL, F.,Ivy
5124N.Willowhaven Drive
Durham,NC27712(US)
(86)PCT/US 2002/000482(en)
(87)WO 2002/053533 11.7.2002
(51) A61K0031/4433 (2006.01) Z C07 D0401/12 (2006.01)
(11) 01562 933
(51) A61K0031/4439 (2006.01) Z C07 D0401/12 (2006.01)
(11) 01562 933
1237
15.4.2008+pat+7
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